产品详情
N-甲基环己基苯并咪唑类似物1; 1-(环己基甲基)-2-[((4-乙氧基苯基)甲基] -N,N-二乙基-1H-苯并咪唑-5-羧酰胺
N-Methylcyclohexyl benzimidazole analog 1; 1-(cyclohexylmethyl)-2-[(4-ethoxyphenyl)methyl]-N,N-diethyl-1H-benzimidazole-5-carboxamide
A potent agonist of the human CB2 receptor (EC50 = 0.52 nM) that shows high selectivity for CB2 over CB1 (Kis = 3.7 and 110 nM, respectively)
背景资料
Several benzimidazole derivatives, developed as synthetic cannabinoid (CB) receptor agonists, have been identified as being selective for the peripheral CB2 receptor.{21225} MCHB-1 is a potent agonist of the human CB2 receptor (EC50 = 0.52 nM) that shows high selectivity for CB2 over CB1 (Kis = 3.7 and 110 nM, respectively).{21225} Similar benzimidazole compounds significantly reduce peripheral pain with reduced central nervous system side effects in mice.{21221} This product is intended for forensic and research applications.
保存条件
建议您在收到Cayman Chemical品牌的MCHB-1 (5 mg)产品后置于-20度保存,产品有效期为730天.
品牌介绍
Cayman Chemical向全球科学工作者提供多研究领域的生化、免疫试剂和分析试剂盒,其产品被广泛应用于肿瘤、氧化氮、神经学、凋亡、氧化性损伤、内分泌学等不同研究领域.Cayman Chemical可提供用于检测的特色试剂盒,如:类花生酸类物质、游离的生物标志、环核苷、激素及氧化氮等;也提供多种高质量试剂,包括:类花生酸类物质、氧化氮试剂及许多相关脂质、脂肪酸、酶和抗体.作为Cayman Chemical在中国的区域总代理,艾美捷科技有限公司将为中国客户提供最全面的Cayman Chemical产品以及客户订制化服务.
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